1. Bobowska, Aneta; Galezowski, Michal; Nowak, Mateusz; Commandeur, Claude; Szeremeta-Spisak, Joanna; Nowogrodzki, Marcin; Obara, Alicja; Dzielak, Anna; Lozinska, Iwona; Dudek, Marcelina; Janiga, Anita; Reus, Jacek; Wronowski, Marek; Zastawna, Magdalena; Radzimierski, Adam; Swirski, Mateusz; Zachmann, Julian; Fabritius, Charles-Henry; Porter, Roderick; Fogt, Joanna Preparation of imidazo[1, 2-a] pyrazines as adenosine A2A receptor modulators for the treatment of various diseases WO 2019002606A1
2. Richards, Gareth; Skerry, Timothy M.; Harrity, Joseph P. A.; Zirimwabagabo, Jean-Olivier; Tozer, Matthew J.; Gibson, Karl Richard; Porter, Roderick Alan; Blaney, Paul Matthew; Glossop, Paul Alan Compounds PCT Int. Appl.(2018), WO2018211275 A1 20181122
3. Svendsen, John Sigurd; Stensen, Wenche; Porter, Roderick Alan Benzothiazole derivatives as dyrk1 inhibitors PCT Int. Appl.(2018), WO2018069468A1 20180419.
4. Alan Ashworth Christopher Lord, Richard Elliott, Dan Niculescu-Duvaz, Roderick Porter, Raymond Boffey, Melanie Bayford, Stuart Firth-Clark, Philip Skone, Ashley Jarvis, Anna Hopkins, Trevor Perrior, Rebekah Key 3-Aryl-5-substituted-isoquinolin-1-one compounds and their therapeutic use WO2015/036759
5. Alan Ashworth Christopher Lord, Richard Elliott, Dan Niculescu-Duvaz, Roderick Porter, Raymond Boffey, Melanie Bayford, Stuart Firth-Clark, , Ashley Jarvis, , Trevor Perrior, Rebekah Key 3-Aryl-5-substituted-isoquinolin-1-one compounds and their therapeutic use PCT/GB2013/050561, WO/2013/132253
6. Richard Blunt, Andrew Eatherton, Mark Healy, James Myatt, Roderick Porter Benzoxazine derivatives as Glycine transport inhibitors PCT/EP2010/062459 WO 2011/023753
7. Richard Blunt, Andrew Eatherton, Mark Healy, James Myatt, Roderick Porter, Benzoxazine derivatives for the treatment of GlyT-1 related disorders PCT/EP2010/062459 WO/2011/012622
8. Roderick Alan Porter Pyrrolidinone derivatives useful for the treatement of psychotic and neurological disorders WO2010018214 A2
9. Roderick Alan Porter Spiroimidazole compounds suitable for the treatment of neurological disorders WO2010018213 A2
10. Cooper David Gwyn, Porter Roderick Alan Compounds which inhibit the glycine transporter and uses thereof in medicine PCT/EP2008/061890 WO2009034062 (A1)
11. Richard Blunt, David Gwyn Cooper, Roderick Alan Porter, Paul Wyman Spiro-condensed imidazolone derivatives inhibiting the glycine transporter WO2009034061
12. Ahmad Nadia Mamoona; Lai, Justine Yeun Quai; Andreotti, Daniele; Marshall, Howard Robert; Nash, David John; Porter, Roderick Alan. Glyt1 transporter inhibitors and uses thereof in treatment of neurological and neuropsychiatric disorders. PCT Int. Appl. (2008), WO 2008092876 A1
13. Coulton, Steven; Porter, Roderick Alan. Glyt1 transporter inhibitors and uses thereof in treatment of neurological and neuropsychiatric disorders. PCT Int. Appl. (2008), WO 2008092872 A1
14. Ahmad, Nadia Mamoona; Jaxa-Chamiec, Albert Andrzej; Lai, Justine Yeun Quai; Porter, Roderick Alan. Glyt1 transporter inhibitors and uses thereof in treatment of neurological and neuropsychiatric disorders. PCT Int. Appl. (2008), WO 2008092873 A1
15. Ahmad, Nadia Mamoona; Lai, Justine Yeun Quai; Marshall, Howard Robert; Nash, David John; Porter, Roderick Alan. Glyt1 transporter inhibitors and uses thereof in treatment of neurological and neuropsychiatric disorders. PCT Int. Appl. (2008), WO 2008092877 A2
16. Coulton, Steven; Gilpin, Martin Leonard; Porter, Roderick Alan. Preparation of aminophenylalkyl benzamides as Glyt1 glycine transporter inhibitors for treatment of psychoses, dementia, or attention deficit disorder. PCT Int. Appl. (2007), WO2007147839 A1
17. Coulton, Steven; Gilpin, Martin Leonard; Porter, Roderick Alan. Preparation of N-[[1-dimethylaminocyclopentyl](phenyl)methyl]-4-fluoro-2-methyl-6-methoxybenzamide as a GlyT1 glycine transporter inhibitor. PCT Int. Appl. (2007), WO2007147836 A1
18. Gentile, Gabriella; Herdon, Hugh Jonathan; Passchier, Johannes; Porter, Roderick Alan. Preparation of radiolabeled aminocyclopentylbenzyl benzamides as ligands for the GlyT1 glycine transporter. PCT Int. Appl. (2007), WO2007147838 A1
19. Coulton, Steven; Gilpin, Martin Leonard; Porter, Roderick Alan. Preparation of aminophenylalkyl benzamides as glycine transporter inhibitors. PCT Int. Appl. (2007), WO2007147834 A1
20. Branch, Clive Leslie; Marshall, Howard; Nash, David John; Porter, Roderick Alan. Preparation of 1-(2-aryl-2-oxoethyl)-3-phenyl-1,4-diazaspiro[4.5]dec-3-en-2-one derivatives as glycine transporter inhibitors. PCT Int. Appl. (2007. WO2007116061
21. Coulton, Steven; Gilpin, Martin; Porter, Roderick Alan. Preparation of (heterocyclic) aminoalkyl benzamides as glycine transporter inhibitors. PCT Int. Appl. (2007), WO2007113309 A2
22. Coulton, Steven; Marshall, Howard; Nash, David John; Porter, Roderick Alan. Preparation of N-phenyl-2-oxo-1,4-diazaspiro[4.5]dec-3-en-1-yl acetamide derivatives as glycine transporter inhibitors. PCT Int. Appl. (2007), WO2007104775 A1
23. Coulton, Steven; Marshall, Howard; Nash, David John; Porter, Roderick Alan. Preparation of N-phenyl-2-oxo-1,4-diazaspiro[4.5]dec-3-en-1-yl acetamide derivatives and their use as glycine transporter inhibitors. PCT Int. Appl. (2007), WO2007104776
24. Branch, Clive Leslie; Marshall, Howard; Mccritchie, Jackie; Porter, Roderick Alan; Spada, Simone. Preparation of N-phenylmethyl heterocyclic amides having activity at the glycine transporter GlyT1. PCT Int. Appl. (2007), WO2007080159
25. Preparation of diazaspirodecenyl- diazaspiroundecenyl- and diazaspirononenyl acetamides as GlyT1 transporter inhibitors for the treatment of psychosis. Dean, Anthony William; Porter, Roderick Alan.. PCT Int. Appl. (2007), WO2007014762 A2
26. Preparation of acylated piperazines as glycine transporter inhibitors. Bradley, Daniel Marcus; Branch, Clive Leslie; Chan, Wai Ngor; Coulton, Steven; Dean, Anthony William; Doyle, Paul Martin; Evans, Brian; Gilpin, Martin Leonard; Gough, Sharon Lisa; Macritchie, Jacqueline Anne; Marshall, Howard Robert; Nash, David John; Porter, Roderick Alan; Ward, Simon Edward. PCT Int. Appl. (2006), WO 2006094842 A1
27. Preparation of N-benzoyl piperazines as glycine transporter inhibitors. Bradley, Daniel Marcus; Branch, Clive Leslie; Brown, Bethany Joy; Chan, Wai Ngor; Coulton, Steven; Dean, Anthony William; Doyle, Paul Martin; Evans, Brian; Gilpin, Martin Leonard; Gough, Sharon Lisa; Macritchie, Jacqueline Anne; Marshall, Howard Robert; Nash, David John; Porter, Roderick Alan; Stasi, Luigi Piero. PCT Int. Appl. (2006), WO 2006094843 A1
28. Preparation of N-( -substituted benzyl) amides as glycine transport inhibitors. Bozzoli, Andrea; Branch, Clive Leslie; Macritchie, Jacqueline Anne; Marshall, Howard Robert; Porter, Roderick Alan; Spada, Simone. PCT Int. Appl. (2006), WO 2006067437 A1
29. Preparation of N-[2-(dimethylamino)-2-methyl-1-phenylpropyl] benzamides as glycine transport inhibitors. Bradley, Daniel Marcus; Branch, Clive Leslie; Chan, Wai Ngor; Coulton, Steven; Gilpin, Martin Leonard; Harris, Andrew Jonathan; Lai, Justine Yeun Quai; Marshall, Howard Robert; Macritchie, Jacqueline Anne; Nash, David John; Porter, Roderick Alan; Spada, Simone; Thewlis, Kevin Michael; Ward, Simon Edward.. PCT Int. Appl. (2006), WO 2006067417 A1
30. Preparation of benzamides as glycine transport inhibitors. Bozzoli, Andrea; Bradley, Daniel Marcus; Coulton, Steven; Gilpin, Martin Leonard; Macritchie, Jacqueline Anne; Porter, Roderick Alan; Thewlis, Kevin Michael. PCT Int. Appl. (2006), WO 2006067414 A2
31. Preparation of N-(phenylmethyl) benzamides as glycine transport inhibitors. Bradley, Daniel Marcus; Branch, Clive Leslie; Chan, Wai Ngor; Coulton, Steven; Gilpin, Martin Leonard; Harris, Andrew Jonathan; Jaxa-Chamiec, Albert Andrzej; Lai, Justine Yeun Quai; Marshall, Howard Robert; Macritchie, Jacqueline Anne; Nash, David John; Porter, Roderick Alan; Spada, Simone; Thewlis, Kevin Michael; Ward, Simon Edward.. PCT Int. Appl. (2006), WO 2006067423 A1
32. Preparation of N-( -substituted benzyl) amides as glycine transport inhibitors. Bozzoli, Andrea; Branch, Clive Leslie; Macritchie, Jacqueline Anne; Marshall, Howard Robert; Porter, Roderick Alan; Spada, Simone. PCT Int. Appl. (2006), WO 2006067430 A1
33. Quinolinecarboxamides having activity at NK3 receptor and their preparations, pharmaceutical compositions and use for treatment of disease mediated by modulation of NK3 receptors. Bradley, Daniel Marcus; Porter, Roderick Alan; Smith, Paul William; Stead, Rachel Elizabeth Anne; Vong, Antonio Kuok Keong.. PCT Int. Appl. (2006), WO 2006050991 A1
34. Preparation of N-morpholinylphenyl-N-(piperidinylmethyl)acetamide derivatives and related compounds as GlyT1 transporter inhibitors for the treatment of mental disorders. Branch, Clive Leslie; Nash, David John; Marshall, Howard; Porter, Roderick Alan.. PCT Int. Appl. (2005), WO 2005103000 A1
35. Preparation of N-morpholinylpyridinyl-N-(piperidinylmethyl)acetamide derivatives and related compounds as GlyT1 transporter inhibitors for the treatment of neurological disorders. Nash, David John; Porter, Roderick Alan.. PCT Int. Appl. (2005), WO 2005103038 A1
36. Preparation of (morpholinyl)phenyl azabicyclooctyl ureas as GlyT1 transporter inhibitors for treating neurological disorders. Bozzoli, Andrea; Branch, Clive Leslie; Marshall, Howard; Nash, David John; Porter, Roderick Alan.. PCT Int. Appl. (2005), WO 2005058317 A1
37. Preparation of (piperidinyl)(morpholinyl)phenyl ureas as GlyT1 transporter inhibitors for treating neurological disorders. Bradley, Daniel Marcus; Branch, Clive Leslie; Marshall, Howard; Nash, David John; Porter, Roderick Alan.. PCT Int. Appl. (2005), 61 pp. WO 2005058885 A2
38. Preparation of compounds having morpholinyl and piperidinyl groups for use as GlyT1 and GlyT2 inhibitors for use in treating neurological disorders. Branch, Clive Leslie; Marshall, Howard; Nash, David John; Porter, Roderick Alan. PCT Int. Appl. (2005), 53 pp. WO 2005058882 A1
39. Preparation of piperidinylhydroxypropylsulfamides as GlyT1 glycine transporter inhibitors for treatment of neurological and neuropsychiatric disorders. Coulton, Steven; Porter, Roderick Alan.. PCT Int. Appl. (2004), WO 2004112787 A1
40. N-(3-Amino-2-hydroxypropyl)benzenesulfonamide derivatives as GlyT1 transporter inhibitors, their preparation, and their use in the treatment of neurological and neuropsychiatric disorders. Branch, Clive Leslie; Nash, David John; Porter, Roderick Alan.. PCT Int. Appl. (2004), WO 2004113280 A1
41. Branch, Clive Leslie; Pilleux, Jean-Pierre; Porter, Roderick Alan. Preparation of tetrahydroquinolines and tetrahydroisoquinolines as orexin receptor antagonists. PCT Int. Appl. (2004), WO 2004041816 A1
42. Coulton, Steven; Porter, Roderick Alan. Preparation of N-(arylsulfonyl) cyclic amines as orexin antagonists. PCT Int. Appl. (2004) WO 2004041807 A1
43. Chan, Wai Ngor; Nash, David John; Porter, Roderick Alan; Stead, Rachel Elizabeth Anne. Preparation of N-(arylacetyl) cyclic amine derivatives as orexin antagonists. PCT Int. Appl. (2004) WO 2004041791 A1
44. Preparation of N-aroyl cyclic amines as orexin receptor antagonists. Branch, Clive Leslie; Coulton, Steven; Johns, Amanda; Nash, David John; Porter, Roderick Alan; Stemp, Geoffrey. (Glaxo Group Limited, UK). PCT Int. Appl. (2004), WO 2004026866 A1
45. Coulton, Steven; Hadley, Michael Stewart; Herdon, Hugh Jonathan; Jin, Jian; Joiner, Graham J.; Porter, Roderick Alan; Rahman, Shahzad Sharooq. Preparation of GlyT1 transporter inhibitors and their use in treatment of neurological and neuropsychiatric disorders. PCT Int. Appl. (2003), WO 2003055478 A1
46. Branch, Clive Leslie; Coulton, Steven; Nash, David John; Porter, Roderick Alan. Preparation of piperazine derivatives as orexin receptor antagonists. PCT Int. Appl. (2003), WO 2003051873 A1
47. Coulton, Steven; Johns, Amanda; Porter, Roderick Alan. Preparation of ethylene diamine derivatives as orexin receptor antagonists. PCT Int. Appl. (2003), WO 2003051872 A1
48. Branch, Clive Leslie; Johns, Amanda; Johnson, Christopher Norbert; Novelli, Riccardo; Porter, Roderick Alan; Stead, Rachel Elizabeth Anne; Stemp, Geoffrey; Thewlis, Kevin. N-aroyl cyclic amine derivatives and their use as orexin receptor antagonist. PCT Int. Appl. (2003), WO 2003051871 A1
49. Chan, Wai Ngor; Johns, Amanda; Porter, Roderick Alan; Stead, Rachel Elizabeth Anne; Vimal, Mythily. Benzamide derivatives as antagonists of orexin receptors. PCT Int. Appl. (2003), WO 2003037847 A1
50. Branch, Clive Leslie; Chan, Wai Ngor; Johns, Amanda; Johnson, Christopher Norbert; Nash, David John; Novelli, Riccardo; Pilleux, Jean-Pierre; Porter, Roderick Alan; Stead, Rachel Elizabeth Anne; Stemp, Geoffrey. Preparation of aroylazoles and aroylazines as orexin receptor antagonists. PCT Int. Appl. (2003), WO 2003002561 A1
51. Chan, Wai Ngor; Johns, Amanda; Johnson, Christopher Norbert; Novelli, Riccardo; Porter, Roderick Alan. Preparation of N-acyl-2-heterocyclyl substituted piperidines and analogs as orexin receptor antagonists. PCT Int. Appl. (2003), WO 2003002559 A2
52. Branch, Clive Leslie; Coulton, Steven; Johns, Amanda; Johnson, Christopher Norbert; Porter, Roderick Alan; Stemp, Geoffrey; Thewlis, Kevin. Preparation of N-aroyl cyclic amines as orexin antagonists. PCT Int. Appl. (2002), WO 2002090355 A1
53. Gaillard, Pascale; Johnson, Christopher Norbert; Novelli, Riccardo; Porter, Roderick Alan; Stemp, Geoffrey; Thewlis, Kevin Michael. Preparation of N-aroyl cyclic amines as orexin receptor antagonists. PCT Int. Appl. (2002), WO 2002089800 A2
54. Novelli, Riccardo; Porter, Roderick Alan. Preparation of condensed tricyclic piperidines having anti-convulsant activity. PCT Int. Appl. (2000), WO 0008023 A1.
55. Coulton, Steven; Porter, Roderick Alan. Preparation of 1-phenyl 3-pyrrolo[2,1-a]isoquinolinyl ureas as anticonvulsants. PCT Int. Appl. (2000), WO 0008022 A1.
56. Coulton, Steven; Novelli, Riccardo; Porter, Roderick Alan; Thompson, Mervyn; Ward, Robert William. Preparation of pyrido[2,1-a]isoquinolines and pyrrolo[2,1-a]isoquinolines as anticonvulsants. PCT Int. Appl. (2000), WO 0008020 A2.
57. Coulton, Steven; Harling, John David; Porter, Roderick Alan; Thompson, Mervyn. Preparation of substituted isoquinolines as anticonvulsants. PCT Int. Appl. (2000), WO 0007993 A1.
58. Coulton, Steven; Johns, Amanda; Porter, Roderick Alan. Preparation of phenyl ureas and thioureas as human orexin receptor antagonists. PCT Int. Appl. (2000), WO 0047580
59. Coulton, Steven; Johns, Amanda; Porter, Roderick Alan. Preparation of phenyl ureas and thioureas as orexin receptor antagonists. PCT Int. Appl. (2000), 45 pp. WO 0047577 A1
60. Johns, Amanda; Porter, Roderick Alan. Preparation of cinnamide derivatives as orexin-1 receptors antagonists. PCT Int. Appl. (2000), WO 0047576 A1.
61. Chan, George; Johns, Amanda; Jurewicz, Anthony; Porter, Roderick Alan; Widdowson, Katherine. Preparation of quinolinylureas and related compounds as HFGAN72 antagonists. PCT Int. Appl. (1999), WO 9909024 A1.
62. Thompson, Mervyn; Porter, Roderick Alan. Preparation of substituted isoquinolinyl ureas as anticonvulsants. PCT Int. Appl. (1999), WO 9914197 A1.
63. Hickey, Deirdre Mary Bernadette; Ife, Robert John; Leach, Colin Andrew; Pinto, Ivan Leo; Porter, Roderick Alan; Smith, Stephen Allan. Preparation of pyrimidinone derivatives as Lp-PLA2 inhibitors. PCT Int. Appl. (1999), WO 9924420 A1.
64. Coulton, Steven; Porter, Roderick Alan; Thompson, Mervyn. Preparation of isoquinoline derivatives as anticonvulsants. PCT Int. Appl. (1999), WO 9925709 A1.
65. Bondinell, William E.; Chan, James; Porter, Roderick A.. Preparation of 3-(4-piperidinyl or 1,2,3,6-tetrahydro-4-pyridinyl)-1H-indol-5-ols for treating a CCR5-mediated diseases. PCT Int. Appl. (1999), WO 9917773 A1.
66. Johns, Amanda; Porter, Roderick Alan. Preparation of naphthyridinylureas and related compounds as orexin A receptor antagonists. PCT Int. Appl. (1999), WO 9958533 A1.
67. Coulton, Steven; Porter, Roderick Alan; Thompson, Mervyn. Preparation of isoquinoline derivatives as anticonvulsants. PCT Int. Appl. (1999), WO 9925709 A1.
68. Thompson, Mervyn; Porter, Roderick Alan. Preparation of substituted isoquinolinyl ureas as anticonvulsants. PCT Int. Appl. (1999), WO 9914197 A1.
69. Kitteringham, John; Porter, Roderick A.; Shipton, Mark R.; Vimal, Mythily; Young, Rodney C.; Borrett, Gary T. Preparation of 3-methyl- and -ethylaminocarbazole-6-carboxamide enantiomers as 5-HT1-like receptor agonists. U.S. (1997), US 5618948.
70. Porter, Roderick Alan. (Pyrimidinyl)piperazines and Their Use as Medicaments. PCT Int. Appl. (1994), WO 9414779 A1.
71. Porter, Roderick Alan; Vimal, Mythily. Preparation of 3-amino-1,2,3,4-tetrahydrocarbazole-6-carboxamides as 5-HT1-like receptor agonists. PCT Int. Appl. (1994), WO 9414773 A1.
72. Borrett, Gary Thomas; Kitteringham, John; Porter, Roderick Alan; Shipton, Mark Ralph; Vimal, Mythily; Young, Rodney Christopher. Enantiomers of carbazole derivatives as 5-HT1-like agonists. PCT Int. Appl. (1994), WO 9414772 A1.
73. Porter, Roderick Alan; Coates, William John. Preparation of tryptamine analogs as 5-HT1-like agonists or partial agonists. PCT Int. Appl. (1994), WO 9414771 A1.
74. Porter, Roderick Alan; Ward, John Gerard. Preparation of tryptamine analogs as 5-HT1-like agonists and partial agonists. PCT Int. Appl. (1994), WO 9414770 A1.
75. Porter, Roderick Alan; Prain, Hunter Douglas; Murray, Kenneth John; Warrington, Brian Herbert. Phenol derivatives as agonists of a cyclic AMP-dependent protein kinase. PCT Int. Appl. (1993), WO 9310107.
76. Porter, Roderick Alan; Prain, Hunter Douglas; Murray, Kenneth John; Warrington, Brian Herbert. Preparation of 5-tetrazolyl-3-pyridinol derivatives and their use as medicaments. PCT Int. Appl. (1993), WO 9310114.
77. Murray, Kenneth John; Porter, Roderick Alan; Prain, Hunter Douglas; Warrington, Brian Herbert. 2-pyridinol derivatives and their use as medicaments. PCT Int. Appl. (1993), WO 9310093 A1.
78. Porter, Roderick Alan; Prain, Hunter Douglas; Murray, Kenneth John; Warrington, Brian Herbert. Pyridinol derivatives as medicaments. PCT Int. Appl. (1993), WO 9307137 A1.
79. Murray, Kenneth John; Porter, Roderick Alan; Warrington, Brian Herbert; Lahouratate, Philippe. Phenol and pyridinol derivatives as lusitropic agents. PCT Int. Appl. (1993), WO 9319754 A1.
80. Porter, Roderick Alan; Murray, Kenneth John; Warrington, Brian Herbert; Prain, Hunter Douglas. Preparation of 6-phenyl-3-(5-tetrazolyl)pyridin-2(H)-one derivatives as cyclic AMP-dependent protein kinase agonists. PCT Int. Appl. (1992), WO 9206085.
81. Murray, Kenneth John; Porter, Roderick Alan; Prain, Hunter Douglas; Warrington, Brian Herbert. Preparation of arylpyridinones as drugs. PCT Int. Appl. (1991), WO 9117987.
82. Manley, Paul W.; Porter, Roderick A.; Lai, Mun F. Preparation of 1-(2-alkenyl)imidazoles as thromboxane synthetase inhibitors. U.S. (1989), US 4837333.
83. Lai, Steve Mun Fook; Manley, Paul William; Porter, Roderick Alan. Alpha-[(phenylmethoxy)methyl]pyridinealkanol derivatives, procedure for their preparation, pharmaceutical composition containing them, and their use. Eur. Pat. Appl. (1988), EP 264114.
84. Lai, Steve Mun Fook; Manley, Paul William; Porter, Roderick Alan. Preparation of -(phenylalkyl)pyridinealkanols as platelet inhibitors. Eur. Pat. Appl. (1988), EP 267439.
85. Manley, Paul William; Porter, Roderick Alan. Preparation and testing of imidazopyridines as platelet-activating factor (PAF) antagonists. Eur. Pat. Appl. (1988), EP 260613.
86. Manley, Paul William; Porter, Roderick Alan; Lai, Mun Fook. Substituted alkenylimidazoles. Eur. Pat. Appl. (1985), EP 150892 A2